SCHEMBL9959487

SCHEMBL9959487

O=C(Nc1cccc(F)c1)C1C(=O)N(O)C(=O)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 2/20 0.42
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9958675 0.86 KMT2A (0.50) HPGDNPC1RAB9AMEN1KMT2A
SCHEMBL31653962 0.86 MEN1 (0.47) RAB9AMEN1KMT2APOLBGAA
SCHEMBL10153609 0.86 MEN1 (0.47) RAB9AMEN1KMT2APOLBGAA
SCHEMBL9959300 0.80 ALDH1A1 (0.42) HTTHPGDNPC1RAB9AMEN1
SCHEMBL9958705 0.76 HDAC4 (0.62) HTTHPGDMEN1KMT2AALDH1A1
SCHEMBL9952811 0.76 MALT1 (0.51) HPGDNPC1RAB9AMEN1KMT2A
SCHEMBL19380274 0.75 HDAC4 (0.44) HTTMEN1KMT2AALDH1A1KDM4E
SCHEMBL31653994 0.75 KCNA5 (0.48) MEN1KMT2APOLBMAPTGAA
SCHEMBL10153606 0.75 KCNA5 (0.48) MEN1KMT2APOLBMAPTGAA
SCHEMBL9953409 0.74 POLB (0.50) RAB9AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO claimed
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed