SCHEMBL9963197

SCHEMBL9963197

CC(C)Oc1cc(C(=O)O)on1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.52
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 2/20 0.38
CHRNA4 P43681 2/20 0.38
SMPD1 P17405 2/20 0.36
GAA P10253 1/20 0.35
PLA2G4A P47712 1/20 0.35
S1PR1 P21453 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
MCL1 Q07820 1/20 0.34
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
S1PR3 Q99500 1/20 0.32
S1PR5 Q9H228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20032117 0.86 SMPD1 (0.36) HCAR2ALDH1A1KMT2ACHRNA4SMPD1
SCHEMBL12667405 0.84 SMPD1 (0.35) HCAR2ALDH1A1CHRNA4SMPD1S1PR1
SCHEMBL26156029 0.83 HCAR2 (0.46) HCAR2CHRNA4SMPD1GAAPLA2G4A
SCHEMBL9963198 0.83 CHRNA4 (0.39) ALDH1A1KMT2ACHRNA4SMPD1SMN1; SMN2
SCHEMBL18739865 0.83 SMPD1 (0.40) HCAR2ALDH1A1CHRNA4SMPD1S1PR1
SCHEMBL23930613 0.82 HCAR2 (0.47) HCAR2CHRNA4SMPD1GAAPLA2G4A
SCHEMBL9963199 0.81 RAB9A (0.48) HCAR2ALDH1A1CHRNA4SMPD1S1PR1
SCHEMBL185759 0.79 HCAR2 (0.57) HCAR2ALDH1A1KMT2ACHRNA4SMPD1
Hydrochloric Acid SCHEMBL2948313 0.78 HCAR2 (0.55) HCAR2ALDH1A1KMT2ACHRNA4SMPD1
SCHEMBL2722839 0.75 HCAR2 (0.52) HCAR2ALDH1A1CHRNA4SMPD1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118251389-A Pyridyl derivatives as sodium channel activators 泽农医药公司 2024-06-25 CN disclosed
US-20230159504-A1 7- OR 8-HYDROXY-ISOQUINOLINE AND 7- OR 8-HYDROXY-QUINOLINE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD) VERTEX PHARMACEUTICALS INCORPORATED 2023-05-25 US disclosed
US-8354403-B2 Pyrrolidine derived beta 3 adrenergic receptor agonists MERCK SHARP & DOHME CORP. (US) 2013-01-15 US disclosed
US-20120157432-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME, CORP. (US) 2012-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120157432-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS ADRB3, ADRB1, ADRB2 HCAR2 315/4885ALDH1A1 534/4885KMT2A 4265/4885
US-20230159504-A1 7- OR 8-HYDROXY-ISOQUINOLINE AND 7- OR 8-HYDROXY-QUINOLINE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD) SERPINA2, SERPINB1, SERPINE1 HCAR2 1639/4885ALDH1A1 542/4885KMT2A 3088/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.