SCHEMBL9965458

SCHEMBL9965458

CC(=O)N1CCC(C(=O)Nc2ccccc2Cc2cc(Cl)cc(Cl)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
POLB P06746 4/20 0.49
MAPK8 P45983 1/20 0.47
MAPK10 P53779 1/20 0.47
TRPV1 Q8NER1 2/20 0.46
HDAC3 O15379 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
ENPP2 Q13822 2/20 0.45
TDP1 Q9NUW8 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CCR3 P51677 1/20 0.44
THRB P10828 1/20 0.44
MGLL Q99685 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9965406 0.84 TRPV1 (0.51) TP53GAAMAPTPOLBTRPV1
SCHEMBL14639698 0.83 TDP1 (0.46) TP53GAAMAPTPOLBTRPV1
SCHEMBL9965381 0.81 POLB (0.53) MAPTPOLBMAPK8MAPK10TRPV1
SCHEMBL642196 0.78 GAA (0.56) TP53GAAPOLBMAPK8MAPK10
SCHEMBL14639718 0.76 GAA (0.48) TP53GAAMAPTPOLBTRPV1
SCHEMBL13028221 0.74 GAA (0.48) TP53GAAMAPTPOLBHDAC3
SCHEMBL9965449 0.74 KDM4E (0.51) MAPTCCR3
SCHEMBL13735120 0.74 HDAC1 (0.65) TP53POLBMAPK8MAPK10HDAC3
SCHEMBL2892697 0.74 KDM4E (0.55) TP53POLBMAPK8MAPK10HDAC3
SCHEMBL9965417 0.74 EPHX2 (0.57) TP53MAPTPOLBMAPK8MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed