SCHEMBL9965464

SCHEMBL9965464

C=C(Nc1ccccc1Oc1cc(Cl)cc(Cl)c1)C1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.45
SLC6A4 P31645 6/20 0.45
SLC6A3 Q01959 6/20 0.45
CXCR2 P25025 4/20 0.45
HTR1A P08908 4/20 0.45
PKM P14618 2/20 0.43
GAA P10253 1/20 0.43
ALDH1A1 P00352 3/20 0.39
NPSR1 Q6W5P4 3/20 0.39
ALOX12 P18054 2/20 0.39
GPR55 Q9Y2T6 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HSP90AB1 P08238 2/20 0.38
TOP2A P11388 2/20 0.38
CYP2D6 P10635 2/20 0.37
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL642234 0.85 GAA (0.62) SLC6A2SLC6A4SLC6A3CXCR2HTR1A
SCHEMBL641983 0.76 GAA (0.66) CXCR2PKMGAAALDH1A1NPSR1
SCHEMBL20463493 0.72 HDAC3 (0.48) GAAMAPTKDM4E
SCHEMBL11158092 0.71 ALDH1A1 (0.52) PKMGAAALDH1A1NPSR1ALOX12
SCHEMBL7974632 0.70 GPR35 (0.50) PKMGAAALDH1A1NPSR1ALOX12
SCHEMBL642196 0.69 GAA (0.56) PKMGAAALDH1A1KMT2AKDM4E
SCHEMBL641183 0.69 GAA (0.53) SLC6A2SLC6A4CXCR2HTR1APKM
SCHEMBL9965467 0.68 HTR2C (0.47) SLC6A2SLC6A4SLC6A3CXCR2HTR1A
SCHEMBL10173892 0.68 GAA (0.54) PKMGAAALDH1A1MEN1KMT2A
SCHEMBL9965415 0.68 ACHE (0.68) PKMGAAALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960347-B1 17-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 3 (17BETA-HSD3) INHIBITORS STERIX LTD (GB) 2012-06-20 EP disclosed