SCHEMBL9966385

SCHEMBL9966385

C=C(/C=C\C(C#N)=C/N)NC(=O)C1(c2ccc(-c3cnc(N)c(CO)c3)cc2)CCOCC1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.44
HDAC1 Q13547 2/20 0.32
BMPR1B O00238 11/20 0.31
BMPR1A P36894 11/20 0.31
TGFBR1 P36897 11/20 0.31
ACVRL1 P37023 11/20 0.31
ACVR1 Q04771 11/20 0.31
KCNH2 Q12809 1/20 0.31
CYP2C9 P11712 1/20 0.31
IDO1 P14902 1/20 0.31
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9966536 0.82 MAP4K4 (0.39) MAP4K4HDAC1CYP2C9
SCHEMBL9936397 0.77 MAP4K4 (0.47) MAP4K4HDAC1KCNH2CYP2C9IDO1
SCHEMBL14295962 0.75 MAP4K4 (0.50) MAP4K4HDAC1BMPR1BBMPR1ATGFBR1
SCHEMBL9966522 0.72 ALOX5AP (0.38)
SCHEMBL9966514 0.71 MAP4K4 (0.40) MAP4K4HDAC1BMPR1BBMPR1ATGFBR1
SCHEMBL9966366 0.71 MAP4K4 (0.46) MAP4K4HDAC1KCNH2CYP2C9
SCHEMBL9966485 0.69 MAP4K4 (0.38) MAP4K4HDAC1CYP2C9MAPK1
SCHEMBL9966458 0.69 GSK3B (0.46) MAP4K4HDAC1CYP2C9
SCHEMBL9940268 0.69 MAP4K4 (0.44) MAP4K4HDAC1
SCHEMBL9966389 0.69 ALOX5 (0.41) MAP4K4HDAC1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082817-A1 BIARYLAMIDE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-21 WO disclosed