SCHEMBL9966536

SCHEMBL9966536

C=C(/C=C\C(=C/N)c1cncc(OC)c1)NC(=O)C1(c2ccc(-c3cnc(N)c(CO)c3)cc2)CCOCC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.39
ALDH1A1 P00352 1/20 0.34
POLB P06746 3/20 0.34
CHEK2 O96017 3/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
HPGD P15428 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
HDAC1 Q13547 1/20 0.31
FYN P06241 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9966385 0.82 MAP4K4 (0.44) MAP4K4CYP2C9HDAC1
SCHEMBL9966458 0.79 GSK3B (0.46) MAP4K4ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL9966457 0.73 RIPK1 (0.40) MAP4K4POLBCHEK2MKNK1MKNK2
SCHEMBL9966366 0.72 MAP4K4 (0.46) MAP4K4ALDH1A1POLBCYP2C9CYP2C19
SCHEMBL9966514 0.72 MAP4K4 (0.40) MAP4K4ALDH1A1HDAC1
SCHEMBL9966389 0.70 ALOX5 (0.41) MAP4K4ALDH1A1MEN1KMT2AHDAC1
SCHEMBL14295962 0.70 MAP4K4 (0.50) MAP4K4ALDH1A1CYP2C9KMT2AHDAC1
SCHEMBL9966380 0.69 PIK3CA (0.33) MAP4K4ALDH1A1HDAC1
SCHEMBL9936397 0.68 MAP4K4 (0.47) MAP4K4CYP2C9HDAC1
SCHEMBL9966360 0.68 GSK3B (0.50) MAP4K4ALDH1A1POLBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082817-A1 BIARYLAMIDE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-21 WO disclosed