SCHEMBL9966514

SCHEMBL9966514

C=C(/C=C\C(=C/N)c1csc(C)n1)NC(=O)C1(c2ccc(-c3cnc(N)c(C)c3)cc2)CCOCC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.40
PIK3CA P42336 3/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
BACE1 P56817 1/20 0.31
BMPR1B O00238 2/20 0.31
BMPR1A P36894 2/20 0.31
TGFBR1 P36897 2/20 0.31
ACVRL1 P37023 2/20 0.31
ACVR1 Q04771 2/20 0.31
PIK3R1 P27986 2/20 0.30
AXL P30530 1/20 0.30
MERTK Q12866 1/20 0.30
MTOR P42345 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9966413 0.88 RIPK1 (0.37) MAP4K4PIK3CAACVR1
SCHEMBL9966449 0.88 MAP4K4 (0.33) MAP4K4USP2ALDH1A1TSHRHSD17B10
SCHEMBL9966365 0.88 USP2 (0.33) MAP4K4USP2ALDH1A1TSHRHSD17B10
SCHEMBL9966486 0.87 MAP4K4 (0.33) MAP4K4USP2ALDH1A1TSHRHSD17B10
SCHEMBL9966380 0.85 PIK3CA (0.33) MAP4K4PIK3CAUSP2ALDH1A1TSHR
SCHEMBL9966308 0.85 ALOX5AP (0.33)
SCHEMBL9966523 0.84 IDO1 (0.36) MAP4K4
SCHEMBL9966562 0.77 MAP4K4 (0.44) MAP4K4PIK3CAUSP2ALDH1A1TSHR
SCHEMBL9966277 0.77 ALOX5AP (0.38)
SCHEMBL9966389 0.73 ALOX5 (0.41) MAP4K4ALDH1A1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082817-A1 BIARYLAMIDE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-21 WO disclosed