SCHEMBL9968571

SCHEMBL9968571

N#Cc1cc(S(=O)(=O)NCc2ccc(O)c(O)c2)ccc1OC(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 4/20 0.43
CYP19A1 P11511 3/20 0.41
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
SCN9A Q15858 7/20 0.39
NAMPT P43490 1/20 0.38
RORC P51449 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9968585 0.84 PKM (0.50) CYP19A1SLC6A2SLC6A4SLC6A3NAMPT
SCHEMBL9968024 0.83 SLC6A2 (0.45) CYP19A1SLC6A2SLC6A4SLC6A3NAMPT
SCHEMBL15609570 0.82 MAPT (0.58)
SCHEMBL9968023 0.81 SLC6A2 (0.41) CYP19A1SLC6A2SLC6A4SLC6A3NAMPT
SCHEMBL9968581 0.81 KDM4E (0.43) CYP19A1SLC6A2SLC6A4SLC6A3NAMPT
SCHEMBL9968569 0.79 MAPK1 (0.44) SLC6A2SLC6A4SLC6A3NAMPT
SCHEMBL9941378 0.76 TSHR (0.58)
SCHEMBL6677829 0.72 SLC22A12 (0.50) SLC22A12
SCHEMBL26536708 0.69 ALDH1A1 (0.52)
SCHEMBL15682729 0.68 MEP1B (0.55) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012082862-A2 ANDROGEN RECEPTOR INHIBITORS AND METHODS OF USE THEREOF BETH ISRAEL DEACONESS MEDICAL CENTER (US) 2012-06-21 WO disclosed