SCHEMBL9968690

SCHEMBL9968690

CC(=O)CCN(C)C(=N)N

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.47
NOS1 P29475 1/20 0.47
NOS2 P35228 1/20 0.47
ALDH1A1 P00352 2/20 0.39
TPSAB1 Q15661 1/20 0.35
PAOX Q6QHF9 2/20 0.33
LMNA P02545 2/20 0.33
SLC15A2 Q16348 1/20 0.33
CHRM1 P11229 1/20 0.33
CA1 P00915 7/20 0.32
CA2 P00918 7/20 0.32
ALOX15 P16050 1/20 0.30
BLM P54132 1/20 0.30
PMP22 Q01453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175734 0.82 NOS3 (0.52) NOS3NOS1NOS2TPSAB1
SCHEMBL4097713 0.77 KMT2A (0.55) NOS3NOS1NOS2ALDH1A1TPSAB1
SCHEMBL430835 0.76
SCHEMBL13804019 0.75 ALDH1A1 (0.47) ALDH1A1PAOXLMNASLC15A2CHRM1
Phosphoric Acid SCHEMBL9074636 0.75 NOS3 (0.46) NOS3NOS1NOS2TPSAB1CA1
SCHEMBL4099423 0.74 NOS3 (0.58) NOS3NOS1NOS2ALDH1A1LMNA
SCHEMBL4093127 0.74 CYP1A2 (0.46) NOS3NOS1NOS2ALDH1A1LMNA
SCHEMBL4093905 0.74 NOS3 (0.45) NOS3NOS1NOS2ALDH1A1TPSAB1
SCHEMBL19133282 0.73 ALDH1A1 (0.45) ALDH1A1PAOXLMNASLC15A2CHRM1
SCHEMBL3360466 0.72 NOS3 (0.43) NOS3NOS1NOS2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8202852-B2 Creatine phosphate analog prodrugs, compositions and uses thereof XENOPORT, INC. (US) 2012-06-19 US disclosed
US-20100137255-A1 CREATINE PHOSPHATE ANALOG PRODRUGS, COMPOSITIONS AND USES THEREOF XENOPORT, INC. (US) 2010-06-03 US disclosed
US-7683043-B2 Membrane permeable; ischemia, heart failure, and neurodegenerative disorders XENOPORT, INC. (US) 2010-03-23 US disclosed
US-20080051371-A1 Membrane permeable; ischemia, heart failure, and neurodegenerative disorders XENOPORT, INC. 2008-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137255-A1 CREATINE PHOSPHATE ANALOG PRODRUGS, COMPOSITIONS AND USES THEREOF CKMT1A; CKMT1B, PYGM, TNNI3 NOS3 2619/4885NOS1 3178/4885NOS2 3005/4885
US-20080051371-A1 Membrane permeable; ischemia, heart failure, and neurodegenerative disorders CKMT1A; CKMT1B, SLC8B1, SLC2A1 NOS3 1610/4885NOS1 2008/4885NOS2 1859/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.