SCHEMBL9971321

SCHEMBL9971321

COc1cc(C(=O)N[C@H]2C(O)O[C@H](CNS(=O)(=O)c3cccc(Cl)c3Cl)C[C@@H]2O)cc(-c2ccc(C#N)cc2)c1

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HK2 P52789 16/20 0.79
HK1 P19367 15/20 0.79
GCK P35557 1/20 0.52
GUSB P08236 1/20 0.36
KAT6A Q92794 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9937898 0.88 HK2 (1.00) HK2HK1GCK
SCHEMBL9937902 0.88 HK2 (1.00) HK2HK1GCK
SCHEMBL9938280 0.66 HK2 (0.76) HK2HK1GCK
SCHEMBL9971340 0.64 HK2 (0.48) HK2HK1GCK
SCHEMBL9971377 0.62 HK2 (0.39) HK2HK1GCK
SCHEMBL9938276 0.62 HK2 (0.75) HK2HK1GCK
SCHEMBL9938814 0.61 HK1 (0.62) HK2HK1GCK
SCHEMBL9938812 0.61 HK1 (0.62) HK2HK1GCK
SCHEMBL9938491 0.59 RXRA (0.64)
SCHEMBL9971339 0.59 HK2 (0.63) HK2HK1GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083145-A1 GLUCOSAMINE DERIVATIVES GLAXO WELLCOME MANUFACTURING PTE LTD (SG) 2012-06-21 WO disclosed