SCHEMBL9987616

SCHEMBL9987616

CC1=CN=C(c2cc(OC(C)C)cc(OC3CCN(S(C)(=O)=O)C3)c2)NC1O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
RORC P51449 2/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
CACNB4 O00305 1/20 0.33
CACNA1A O00555 1/20 0.33
CACNA1G O43497 1/20 0.33
CACNG3 O60359 1/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1H O95180 1/20 0.33
CACNB3 P54284 1/20 0.33
CACNA2D1 P54289 1/20 0.33
CACNG7 P62955 1/20 0.33
CACNA1B Q00975 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNB1 Q02641 1/20 0.33
CACNG1 Q06432 1/20 0.33
CACNB2 Q08289 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9987614 0.74 KDM4E (0.38) KDM4ERORCPDE4APDE4BPDE4C
SCHEMBL9987406 0.74 GCK (0.56) KDM4ERORCPDE4APDE4BPDE4C
SCHEMBL9987668 0.73 RORC (0.46) KDM4ERORCCACNB4CACNA1ACACNA1G
SCHEMBL9986894 0.73 KDM4E (0.47) KDM4ERORCPDE4APDE4BPDE4C
SCHEMBL9987288 0.73 GCK (0.56) KDM4ELRRK2
SCHEMBL1140554 0.68 KDM4E (0.48) KDM4ERORCCACNB4CACNA1ACACNA1G
SCHEMBL1107306 0.67 KDM4E (0.47) KDM4ERORCCACNB4CACNA1ACACNA1G
SCHEMBL15263144 0.65 HRH3 (0.43) RORCPDE4APDE4BPDE4CPDE4D
SCHEMBL15263145 0.65 HRH3 (0.43) RORCPDE4APDE4BPDE4CPDE4D
SCHEMBL15428503 0.65 HRH3 (0.43) RORCPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011158149-A1 2-(3,5-DISUBSTITUTEDPHENYL)PYRIMIDIN-4(3H)-ONE DERIVATIVES PFIZER INC. (US) 2011-12-22 WO disclosed