SCHEMBL9987668

SCHEMBL9987668

CC(C)Oc1cc(C#N)cc(OC2CCN(S(C)(=O)=O)C2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 5/20 0.46
RORA P35398 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HRH3 Q9Y5N1 8/20 0.41
FPR2 P25090 1/20 0.39
PROKR1 Q8TCW9 1/20 0.39
CYP2D6 P10635 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALK Q9UM73 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
CACNB4 O00305 1/20 0.35
CACNA1A O00555 1/20 0.35
CACNA1G O43497 1/20 0.35
CACNG3 O60359 1/20 0.35
CACNA1F O60840 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNB3 P54284 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9986894 0.83 KDM4E (0.47) RORCKDM4EHRH3CYP2D6MEN1
SCHEMBL1140554 0.78 KDM4E (0.48) RORCRORAKDM4EHRH3CYP2D6
SCHEMBL1107306 0.77 KDM4E (0.47) RORCRORAKDM4EHRH3CYP2D6
SCHEMBL9987288 0.75 GCK (0.56) KDM4E
SCHEMBL9987614 0.74 KDM4E (0.38) RORCKDM4EHRH3FPR2PROKR1
SCHEMBL9987406 0.74 GCK (0.56) RORCKDM4ECACNB4CACNA1ACACNA1G
SCHEMBL9987616 0.73 KDM4E (0.37) RORCKDM4EHRH3FPR2PROKR1
SCHEMBL15428503 0.71 HRH3 (0.43) RORCHRH3FPR2PROKR1CYP2D6
SCHEMBL15263145 0.71 HRH3 (0.43) RORCHRH3FPR2PROKR1CYP2D6
SCHEMBL18672933 0.71 RORC (0.53) RORCRORAHRH3FPR2PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011158149-A1 2-(3,5-DISUBSTITUTEDPHENYL)PYRIMIDIN-4(3H)-ONE DERIVATIVES PFIZER INC. (US) 2011-12-22 WO disclosed