SCHEMBL9988915

SCHEMBL9988915

COc1cccc(-c2cc(CCC(=O)NCc3cccc(C)n3)nn2-c2ccc(F)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
SLC16A3 O15427 9/20 0.46
SLC16A1 P53985 9/20 0.46
MCTS1 Q9ULC4 3/20 0.46
MALT1 Q9UDY8 1/20 0.45
RXRA P19793 2/20 0.44
RXRB P28702 2/20 0.44
RXRG P48443 2/20 0.44
ALDH1A1 P00352 2/20 0.43
ALOX5 P09917 1/20 0.42
PTGS2 P35354 1/20 0.42
CCKAR P32238 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9989142 0.86 CA1 (0.48) CA1CA2CA9SLC16A3SLC16A1
SCHEMBL9988456 0.86 SLC16A3 (0.53) CA1CA2CA9SLC16A3SLC16A1
SCHEMBL9989540 0.84 MALT1 (0.52) CA1CA2CA9SLC16A3SLC16A1
SCHEMBL9988484 0.84 MALT1 (0.47) MALT1RXRARXRBRXRGALDH1A1
SCHEMBL9989408 0.80 DRD4 (0.51) CA1CA2CA9SLC16A3SLC16A1
SCHEMBL9988534 0.80 MALT1 (0.55) MALT1RXRARXRBRXRGALDH1A1
SCHEMBL9990073 0.80 RXRA (0.48) CA1CA2CA9SLC16A3SLC16A1
SCHEMBL9989046 0.80 TP53 (0.50) SLC16A3SLC16A1MCTS1MALT1RXRA
SCHEMBL9990141 0.79 RXRA (0.51) CA1CA2CA9SLC16A3SLC16A1
SCHEMBL9988387 0.79 DRD4 (0.49) CA1CA2CA9PTGS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011161615-A1 5-LIPOXYGENASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2011-12-29 WO disclosed