SCHEMBL9995252

SCHEMBL9995252

CON(CCN1CCCC1)C(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KMT2A Q03164 3/20 0.50
GFER P55789 1/20 0.49
HRH3 Q9Y5N1 4/20 0.47
SIGMAR1 Q99720 2/20 0.47
LTA4H P09960 1/20 0.47
DRD2 P14416 1/20 0.45
DRD1 P21728 1/20 0.45
DRD3 P35462 1/20 0.45
PTGIR P43119 2/20 0.44
KDM4E B2RXH2 2/20 0.44
HRH4 Q9H3N8 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
MCHR1 Q99705 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15825900 0.90 DRD2 (0.47) ALDH1A1HRH3DRD2PTGIR
SCHEMBL5147435 0.81 HRH3 (0.60) ALDH1A1KMT2AGFERHRH3SIGMAR1
SCHEMBL7251010 0.78 ALDH1A1 (0.58) ALDH1A1KMT2AGFERHRH3SIGMAR1
SCHEMBL3038951 0.75 HPGD (0.44) ALDH1A1KMT2AKDM4E
SCHEMBL28557449 0.73 HPGD (0.47) ALDH1A1
SCHEMBL4518449 0.73 HTT (0.44) ALDH1A1KMT2A
SCHEMBL2796840 0.72 TSHR (0.44) ALDH1A1KMT2AKDM4E
SCHEMBL7244646 0.71 NPC1 (0.49) ALDH1A1KMT2AHRH3SIGMAR1LTA4H
SCHEMBL3066309 0.71 KDM4E (0.55) ALDH1A1KMT2AHRH3KDM4EHRH4
SCHEMBL4930913 0.71 SIGMAR1 (0.50) HRH3SIGMAR1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585470-A2 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHD3ITION OF TYROSINE KINASE ACTIVITY Hanmi Science Co., Ltd. (KR) 2013-05-01 EP disclosed
WO-2011162515-A2 NOVEL FUSED PYRIMIDINE DERIVATIVES FOR INHD3ITION OF TYROSINE KINASE ACTIVITY HANMI HOLDINGS CO. , LTD. (KR) 2011-12-29 WO disclosed