SCHEMBL5147435

SCHEMBL5147435

CN(CCN1CCCC1)C(=O)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.60
ALDH1A1 P00352 3/20 0.54
KMT2A Q03164 3/20 0.54
SIGMAR1 Q99720 2/20 0.53
ACHE P22303 1/20 0.53
TACR2 P21452 1/20 0.53
GFER P55789 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24569593 0.87 OPRD1 (0.50) HRH3SIGMAR1ACHE
SCHEMBL28037481 0.87 ALDH1A1 (0.58) HRH3ALDH1A1KMT2AACHE
SCHEMBL14174804 0.85 NPSR1 (0.52) HRH3ALDH1A1KMT2ASIGMAR1
SCHEMBL16565552 0.84 KDM4E (0.51) HRH3ALDH1A1ACHE
SCHEMBL7251010 0.81 ALDH1A1 (0.58) HRH3ALDH1A1KMT2ASIGMAR1GFER
SCHEMBL15742584 0.81 SIGMAR1 (0.46) HRH3SIGMAR1
SCHEMBL16565555 0.81 ALDH1A1 (0.50) HRH3ALDH1A1KMT2AACHE
SCHEMBL9995252 0.81 ALDH1A1 (0.50) HRH3ALDH1A1KMT2ASIGMAR1GFER
SCHEMBL10149206 0.80 DRD4 (0.53) HRH3ALDH1A1KMT2ASIGMAR1
SCHEMBL11210779 0.79 KMT2A (0.56) ALDH1A1KMT2AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108473478-A TBK/IKK inhibitor compounds and uses thereof 默克专利有限公司 2018-08-31 CN disclosed
EP-1809614-A2 BENZOTRIAZINE INHIBITORS OF KINASES Targegen, Inc. (US) 2007-07-25 EP disclosed
WO-2005096784-A2 BENZOTRIAZINE INHIBITORS OF KINASES TARGEGEN, INC. (US) 2005-10-20 WO disclosed