SCHEMBL9998442

SCHEMBL9998442

CC(CN1CCN(c2ncccn2)CC1)NC(=O)CCc1nc(-c2ccccc2)c(-c2ccccc2)o1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 3/20 0.54
KDM4E B2RXH2 1/20 0.48
ABCC4 O15439 1/20 0.48
C5 P01031 1/20 0.48
LMNA P02545 1/20 0.48
CHRM2 P08172 1/20 0.48
CYP3A4 P08684 1/20 0.48
CHRM1 P11229 1/20 0.48
DRD2 P14416 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
RXRA P19793 1/20 0.48
TBXA2R P21731 1/20 0.48
NR4A1 P22736 1/20 0.48
PTGS1 P23219 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
MAPK1 P28482 1/20 0.48
RXRB P28702 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766610 0.82 NR4A2 (0.54) NR4A2KDM4EABCC4C5LMNA
SCHEMBL9998261 0.77 MAPT (0.49)
SCHEMBL9998326 0.75 KDM4E (0.48) KDM4EHPGD
SCHEMBL4498016 0.73 MEN1 (0.52) KDM4EHPGDCYP2C19
SCHEMBL9998826 0.73 MEN1 (0.52) KDM4EHPGDCYP2C19
Oxaprozin SCHEMBL20657782 0.72 LMNA (0.61) NR4A2KDM4EABCC4C5LMNA
SCHEMBL21675691 0.72 NR4A2 (1.00) NR4A2KDM4EABCC4C5LMNA
SCHEMBL31582641 0.70 NR4A2 (0.77) NR4A2KDM4EABCC4C5LMNA
SCHEMBL21675690 0.70 NR4A2 (0.76) NR4A2KDM4EABCC4C5LMNA
SCHEMBL17208133 0.70 RXRA (0.72) NR4A2KDM4EABCC4C5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917262-B1 PIPERIDINE AND PIPERAZINE DERIVATIVES AS P2X3 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-12-14 EP disclosed