SCHEMBL9998455

SCHEMBL9998455

CC(=O)OCC(=Cc1cccc(Br)c1)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
HTT P42858 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
HSD17B3 P37058 1/20 0.42
SLC6A19 Q695T7 1/20 0.41
ALDH1A1 P00352 2/20 0.40
BACE1 P56817 1/20 0.38
HSD17B10 Q99714 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MCL1 Q07820 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9997664 0.84 LMNA (0.44) PKMMEN1KMT2AALDH1A1POLB
SCHEMBL9998151 0.84 PKM (0.48) PKMHTTMEN1KMT2AAKR1C3
SCHEMBL9998153 0.84 PKM (0.48) PKMHTTMEN1KMT2AAKR1C3
SCHEMBL9998284 0.83 MAPT (0.48) MEN1KMT2AAKR1C3AKR1C2ALDH1A1
SCHEMBL9997762 0.83 PPARG (0.37) HTTMEN1KMT2AALDH1A1MAPT
SCHEMBL9998221 0.83 FBP1 (0.44) PKMMEN1KMT2AAKR1C3ALDH1A1
SCHEMBL9997578 0.82 KMT2A (0.49) PKMHTTMEN1KMT2AAKR1C3
SCHEMBL9998219 0.82 HDAC4 (0.39) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL9998202 0.82 MEN1 (0.47) HTTMEN1KMT2AAKR1C3ALDH1A1
SCHEMBL9997678 0.81 ACHE (0.38) HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8558012-B2 2-fluoro-1,3-benzodithiol 1,1,3,3-tetraoxide derivative, production method thereof, and production method of monofluoromethyl group-containing compound using the same NAGOYA INSTITUTE OF TECHNOLOGY (JP) 2013-10-15 US disclosed
US-20110319637-A1 2-FLUORO-1,3-BENZODITHIOL 1,1,3,3-TETRAOXIDE DERIVATIVE, PRODUCTION METHOD THEREOF, AND PRODUCTION METHOD OF MONOFLUOROMETHYL GROUP-CONTAINING COMPOUND USING THE SAME NAGOYA INSTITUTE OF TECHNOLOGY (JP) 2011-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110319637-A1 2-FLUORO-1,3-BENZODITHIOL 1,1,3,3-TETRAOXIDE DERIVATIVE, PRODUCTION METHOD THEREOF, AND PRODUCTION METHOD OF MONOFLUOROMETHYL GROUP-CONTAINING COMPOUND USING THE SAME CBR1, CYP1B1, CYP2F1 PKM 1948/4885HTT 1667/4885MEN1 1032/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.