SCHEMBL9998646

SCHEMBL9998646

Cc1cccc(C(C(=O)O)N2CN(c3ccccc3)C3(CCNCC3)C2=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.46
OPRD1 P41143 9/20 0.46
OPRK1 P41145 9/20 0.46
OPRL1 P41146 9/20 0.46
ENPP2 Q13822 3/20 0.41
HSD17B10 Q99714 1/20 0.40
DDR1 Q08345 2/20 0.38
BDKRB2 P30411 1/20 0.37
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
PLD2 O14939 1/20 0.36
PLD1 Q13393 1/20 0.36
NPC1L1 Q9UHC9 1/20 0.36
METAP2 P50579 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9998330 0.87 OPRM1 (0.44) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL9998993 0.83 OPRL1 (0.45) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL10248464 0.83 OPRK1 (0.51) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL10248209 0.83 OPRK1 (0.51) OPRM1OPRD1OPRK1OPRL1HSD17B10
Toluene SCHEMBL318509 0.81 OPRM1 (0.43) OPRM1OPRD1OPRK1OPRL1ENPP2
SCHEMBL318086 0.80 OPRL1 (0.48) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL318087 0.80 OPRL1 (0.48) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL318391 0.80 OPRL1 (0.48) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL318533 0.78 OPRM1 (0.46) OPRM1OPRD1OPRK1OPRL1HSD17B10
SCHEMBL318548 0.78 OPRM1 (0.46) OPRM1OPRD1OPRK1OPRL1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2582701-A1 D2 ANTAGONISTS, METHODS OF SYNTHESIS AND METHODS OF USE Altos Therapeutics, LLC (US) 2013-04-24 EP disclosed
WO-2011160084-A1 D2 ANTAGONISTS, METHODS OF SYNTHESIS AND METHODS OF USE Altos Therapeutics, LLC (US) 2011-12-22 WO disclosed