SCHEMBL10033100

SCHEMBL10033100

CCOC(=O)CC1CCCC(N)C1c1cc(F)c(F)cc1F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
ALDH1A1 P00352 4/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
PPOX P50336 1/20 0.32
KDM4E B2RXH2 2/20 0.31
TSHR P16473 1/20 0.31
ITGB3 P05106 2/20 0.31
ITGA2B P08514 2/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
DPP4 P27487 2/20 0.31
DPP9 Q86TI2 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033129 0.88 PPOX (0.36) CYP11B1CYP11B2ALDH1A1ALOX5APFEN1
SCHEMBL10033128 0.87 ALOX5AP (0.36) CYP11B1CYP11B2ALDH1A1ALOX5APFEN1
SCHEMBL10033112 0.85 BRD4 (0.42) ALDH1A1ALOX5APFEN1KDM4ETSHR
SCHEMBL10033098 0.84 ALOX5AP (0.39) CYP11B1CYP11B2ALDH1A1ALOX5APFEN1
SCHEMBL10033106 0.81 HTR2A (0.38) CYP11B1CYP11B2ALDH1A1ALOX5APFEN1
SCHEMBL10033113 0.81 L3MBTL1 (0.42) CYP11B1CYP11B2ALDH1A1ALOX5APFEN1
SCHEMBL10033104 0.80 MEN1 (0.38) ALDH1A1L3MBTL1KDM4EMAPK1NPSR1
SCHEMBL10033095 0.79 L3MBTL1 (0.41) ALDH1A1ALOX5APFEN1L3MBTL1PPOX
SCHEMBL12418257 0.76 GAA (0.39) ALDH1A1L3MBTL1POLBCYP1A2
SCHEMBL10033130 0.74 TACR1 (0.41) CYP11B1CYP11B2ALDH1A1KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed