SCHEMBL10033112

SCHEMBL10033112

CCOC(=O)CC1CCCC(N)C1c1ccccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.42
ALDH1A1 P00352 5/20 0.41
CYP1A2 P05177 2/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TSHR P16473 3/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
BCHE P06276 1/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NLRP3 Q96P20 1/20 0.36
IDO1 P14902 1/20 0.35
KDM1A O60341 3/20 0.35
KDM1B Q8NB78 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033128 0.86 ALOX5AP (0.36) BRD4ALDH1A1MAPK1NPSR1TSHR
SCHEMBL10033098 0.85 ALOX5AP (0.39) ALDH1A1MAPK1NPSR1TSHRHSD17B10
SCHEMBL10033100 0.85 CYP11B1 (0.35) ALDH1A1CYP1A2MAPK1NPSR1TSHR
SCHEMBL10033104 0.81 MEN1 (0.38) ALDH1A1CYP1A2MAPK1NPSR1HSD17B10
SCHEMBL10033129 0.80 PPOX (0.36) ALDH1A1TSHRKMT2AKDM4EPOLB
SCHEMBL10033106 0.80 HTR2A (0.38) ALDH1A1MAPK1TSHRHSD17B10KMT2A
SCHEMBL10033113 0.80 L3MBTL1 (0.42) ALDH1A1TSHRSMN1; SMN2KDM1AALOX5AP
SCHEMBL10033182 0.78 BRD4 (0.38) BRD4ALDH1A1CYP1A2TSHRKDM4E
SCHEMBL10033095 0.78 L3MBTL1 (0.41) ALDH1A1NPSR1KMT2ASMN1; SMN2ALOX5AP
SCHEMBL10033130 0.76 TACR1 (0.41) ALDH1A1MAPK1NPSR1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed