SCHEMBL10038837

SCHEMBL10038837

CCOC(=O)Cc1c(C)nc2ccc(CC)cn12

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC2A2 P11168 1/20 0.49
MAPK1 P28482 1/20 0.44
GAA P10253 1/20 0.41
KDM4E B2RXH2 3/20 0.41
RXFP1 Q9HBX9 2/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
CYP4Z1 Q86W10 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12017652 0.88 SLC2A2 (0.46) SLC2A2MAPK1GAAKDM4ERXFP1
SCHEMBL10038836 0.84 ALDH1A1 (0.39) MAPK1GAAKDM4EKMT2ARAB9A
SCHEMBL3594242 0.79 SLC2A2 (0.46) SLC2A2MAPK1GAANPC1RAB9A
SCHEMBL13500447 0.76 MAPK1 (0.50) MAPK1GAAKDM4ERXFP1KMT2A
SCHEMBL2260441 0.76 KDM4E (0.47) SLC2A2GAAKDM4ERXFP1KMT2A
SCHEMBL16115202 0.74 SLC2A2 (0.47) SLC2A2GAAKDM4ERXFP1MAPT
SCHEMBL3594244 0.72 SLC2A2 (0.46) SLC2A2MAPK1GAAKDM4ENPC1
SCHEMBL27500927 0.72 GABRA1 (0.72) SLC2A2KDM4ENPC1RAB9A
SCHEMBL23624072 0.70 SLC2A2 (0.82) SLC2A2MAPK1GAAKDM4EMAPT
SCHEMBL10299459 0.69 CYP4Z1 (0.57) MAPK1GAAKDM4EKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193236-B2 Indolylmaleimide derivatives processes for their production and pharmaceutical compositions NOVARTIS AG (CH) 2012-06-05 US disclosed
US-20100041693-A1 INDOLYLMALEIMIDE DERIVATIVES NOVARTIS AG (CH) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041693-A1 INDOLYLMALEIMIDE DERIVATIVES IDH3A, IDH2, INMT SLC2A2 2956/4885MAPK1 3536/4885GAA 2381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.