SCHEMBL10040299

SCHEMBL10040299

O=c1ccc(-c2cccc(C(F)(F)F)c2)nn1C1CC=NN1c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
LMNA P02545 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HDAC1 Q13547 1/20 0.38
KDM1A O60341 3/20 0.38
MAOB P27338 2/20 0.37
KMT2A Q03164 1/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14973530 0.68 ALDH1A1 (0.50) ALDH1A1LMNANPSR1HPGDKDM4E
SCHEMBL6697417 0.66 ALDH1A1 (0.66) ALDH1A1LMNANPSR1HPGDKDM4E
SCHEMBL4723906 0.65 HDAC1 (0.51) ALDH1A1LMNANPSR1HPGDKDM4E
SCHEMBL10039579 0.64 AADAT (0.43) ALDH1A1HPGDCYP1A2CYP3A4KDM1A
SCHEMBL8103915 0.63 CTSS (0.60)
SCHEMBL8102136 0.62 CTSS (0.67)
SCHEMBL9229195 0.62 NPSR1 (1.00) ALDH1A1LMNANPSR1KDM4ECYP1A2
SCHEMBL4721881 0.62 GAA (0.43) ALDH1A1LMNANPSR1HPGDKDM4E
SCHEMBL19657972 0.61 ALDH1A1 (0.70) ALDH1A1LMNANPSR1HPGDCYP1A2
SCHEMBL16474677 0.60 HTT (0.49) ALDH1A1LMNANPSR1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020780-A1 HETEROCYCLIC COMPOUND AND USE THEREOF 武田薬品工業株式会社 (JP) 2012-02-16 WO disclosed