SCHEMBL10054559

SCHEMBL10054559

COc1ccc(CN2CCC3CNCCC32)cc1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.44
REN P00797 2/20 0.43
HTR1A P08908 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
HRH1 P35367 2/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053945 0.82 HTR1A (0.45) SIGMAR1HTR1A
SCHEMBL18618012 0.77 HRH2 (0.46) SIGMAR1
SCHEMBL3648634 0.76 CHRNB2 (0.47) SIGMAR1REN
SCHEMBL3650270 0.76 CHRNB2 (0.47) SIGMAR1REN
Hydrochloric Acid SCHEMBL4537169 0.75 SIGMAR1 (0.47) SIGMAR1REN
SCHEMBL17606834 0.74 LTA4H (0.44) SIGMAR1CYP3A4CYP2D6
SCHEMBL28496997 0.73 HRH2 (0.56) SIGMAR1
SCHEMBL28231989 0.73 SIGMAR1 (0.46) SIGMAR1
SCHEMBL30775094 0.73 SIGMAR1 (0.55) SIGMAR1
SCHEMBL28148266 0.73 HSD11B1 (0.46) SIGMAR1CYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019426-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed