SCHEMBL100652

SCHEMBL100652

CC(C)(C)[Si](C)(C)OCc1ccc(NC(=O)CCc2ccc(-c3ccccc3)c(NC(=O)O)c2)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 11/20 0.44
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
LTB4R Q15722 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL102617 0.95 HCAR2 (0.39) HCAR2NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL101458 0.91 HCAR2 (0.45) HCAR2RAB9AMEN1KMT2AAKR1C3
SCHEMBL102082 0.90 RAB9A (0.44) HCAR2NPC1RAB9ASMN1; SMN2AKR1C3
SCHEMBL102147 0.89 LTB4R (0.44) HCAR2HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL98766 0.88 LTB4R (0.52) HCAR2HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL99813 0.87 HCAR2 (0.44) HCAR2RAB9A
SCHEMBL100322 0.87 HPGD (0.44) HCAR2NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL101812 0.85 PTGDR2 (0.42) HCAR2NPC1RAB9A
SCHEMBL99078 0.85 HCAR2 (0.42) HCAR2RAB9AHPGDMEN1KMT2A
SCHEMBL663614 0.85 CHRM3 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed