SCHEMBL101458

SCHEMBL101458

Cc1cc(CO[Si](C)(C)C(C)(C)C)ccc1NC(=O)CCc1ccc(-c2ccccc2)c(NC(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 10/20 0.45
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.39
LTB4R Q15722 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL100652 0.91 HCAR2 (0.44) HCAR2MEN1KMT2AAKR1C3AKR1C2
SCHEMBL102082 0.91 RAB9A (0.44) HCAR2AKR1C3AKR1C2RAB9ALTB4R
SCHEMBL102147 0.90 LTB4R (0.44) HCAR2MEN1KMT2AMAPTLTB4R
SCHEMBL98766 0.89 LTB4R (0.52) HCAR2MEN1KMT2AMAPTLTB4R
SCHEMBL99813 0.89 HCAR2 (0.44) HCAR2HTTRAB9AMAPT
SCHEMBL99078 0.87 HCAR2 (0.42) HCAR2MEN1KMT2ALMNAHTT
SCHEMBL99712 0.86 HDAC1 (0.40) HCAR2MEN1KMT2ALMNAL3MBTL1
SCHEMBL100027 0.86 GAA (0.39) HCAR2MEN1KMT2AGAALMNA
SCHEMBL102617 0.86 HCAR2 (0.39) HCAR2MEN1KMT2ARAB9APOLB
SCHEMBL99669 0.86 NPC1 (0.45) HCAR2MEN1KMT2ARAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed