SCHEMBL10068544

SCHEMBL10068544

COC(=O)c1cc(OCC(F)(F)F)cc(C(O)c2cccc(Cl)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.43
ADRB3 P13945 4/20 0.43
ADRB2 P07550 3/20 0.43
MRGPRX4 Q96LA9 4/20 0.42
BRD4 O60885 1/20 0.41
CREBBP Q92793 1/20 0.41
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.37
S1PR2 O95136 1/20 0.37
S1PR4 O95977 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
XBP1 P17861 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
PAX8 Q06710 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
S1PR3 Q99500 1/20 0.37
S1PR5 Q9H228 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10068720 0.87 BRD4 (0.53) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10068778 0.85 HPGD (0.43) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10068557 0.85 BRD4 (0.42) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10069315 0.84 ADRB1 (0.43) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10068770 0.84 FAAH (0.44) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10068957 0.84 HPGD (0.42) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10069563 0.83 ADRB2 (0.47) ADRB1ADRB3ADRB2MEN1MAPT
SCHEMBL10068568 0.82 SMN1; SMN2 (0.45) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10068804 0.82 F2 (0.43) ADRB1ADRB3ADRB2BRD4CREBBP
SCHEMBL10068545 0.81 ADRB2 (0.37) ADRB1ADRB3ADRB2MRGPRX4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958912-B Benzohydrol derivatives, a preparation process and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2015-01-14 CN disclosed
WO-2012019428-A1 BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed