SCHEMBL10068804

SCHEMBL10068804

COC(=O)c1cc(OCC2CC2)cc(C(O)c2cccc(Cl)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.43
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
FFAR1 O14842 9/20 0.41
CNR2 P34972 1/20 0.40
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
ACACA Q13085 2/20 0.39
GPR88 Q9GZN0 1/20 0.39
ACACB O00763 1/20 0.39
NR1H4 Q96RI1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10068720 0.86 BRD4 (0.53) BRD4CREBBPADRB2ADRB1ADRB3
SCHEMBL10068778 0.84 HPGD (0.43) BRD4CREBBPADRB2ADRB1ADRB3
SCHEMBL10068557 0.84 BRD4 (0.42) BRD4CREBBPADRB2ADRB1ADRB3
SCHEMBL10069315 0.83 ADRB1 (0.43) BRD4CREBBPADRB2ADRB1ADRB3
SCHEMBL10068770 0.83 FAAH (0.44) BRD4CREBBPADRB2ADRB1ADRB3
SCHEMBL10068957 0.83 HPGD (0.42) BRD4CREBBPFFAR1ADRB2ADRB1
SCHEMBL10068544 0.82 ADRB1 (0.43) BRD4CREBBPADRB2ADRB1ADRB3
SCHEMBL10069563 0.82 ADRB2 (0.47) ADRB2ADRB1ADRB3
SCHEMBL10068801 0.81 REN (0.41) F2FFAR1CNR2
SCHEMBL10069336 0.79 SLC6A3 (0.43) ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958912-B Benzohydrol derivatives, a preparation process and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2015-01-14 CN disclosed
WO-2012019428-A1 BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed