SCHEMBL10070046

SCHEMBL10070046

CCCCOc1c(C(=O)O)nc2c(N(C)S(C)(=O)=O)cc(Br)cn2c1=O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
THRA P10827 3/20 0.33
THRB P10828 3/20 0.33
MMP9 P14780 2/20 0.32
MMP2 P08253 1/20 0.32
CYP19A1 P11511 2/20 0.32
CNR2 P34972 1/20 0.32
MMP1 P03956 1/20 0.31
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10070944 0.91 MMP9 (0.34) THRATHRBMMP9MMP2CYP19A1
SCHEMBL10070392 0.81 TLR7 (0.30)
SCHEMBL12894144 0.74 MAPT (0.36) KDM4E
SCHEMBL15101373 0.73 MET (0.30)
SCHEMBL10069877 0.71 THRA (0.34) THRATHRBCNR2LMNA
SCHEMBL10071002 0.70 TSHR (0.36) THRATHRBCNR2LMNAKDM4E
SCHEMBL12894051 0.69 MAPT (0.39) THRATHRBLMNAKDM4E
SCHEMBL10070414 0.69 CNR2 (0.39) CNR2
SCHEMBL12140417 0.67 MAPT (0.39) THRBLMNAKDM4E
SCHEMBL10071008 0.66 ALDH1A1 (0.33) MMP9MMP1MMP13ADAM17LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006680-A1 7, 9-NITROGEN RADICAL-4-OXO-4H-PYRIDO[L,2-A]PYRIMIDINE-2-CARBOXYLIC ACID BENZYLAMIDE ANTI-VIRALS AVEXA LIMITED (AU) 2012-01-19 WO disclosed