SCHEMBL10072044

SCHEMBL10072044

Cc1ccc2ncnc(N3CCOc4ccccc43)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.44
MAPK1 P28482 5/20 0.43
ALDH1A1 P00352 5/20 0.43
CLK4 Q9HAZ1 5/20 0.43
HIF1A Q16665 4/20 0.43
CYP2C19 P33261 3/20 0.43
TSHR P16473 3/20 0.43
CSF1R P07333 1/20 0.43
NUDT1 P36639 1/20 0.43
CHRM4 P08173 1/20 0.41
PDGFRB P09619 2/20 0.41
LMNA P02545 3/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
USP2 O75604 2/20 0.41
CYP2D6 P10635 1/20 0.41
KDM4E B2RXH2 2/20 0.40
HTT P42858 2/20 0.40
PDE5A O76074 1/20 0.40
KDR P35968 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10072046 0.87 NUDT1 (0.42) EGFRMAPK1ALDH1A1CLK4HIF1A
SCHEMBL14595182 0.72 ALDH1A1 (0.65) MAPK1ALDH1A1CLK4HIF1ACYP2C19
SCHEMBL3805071 0.72 LMNA (0.54) MAPK1ALDH1A1TSHRCHRM4LMNA
SCHEMBL171792 0.71 NOTUM (0.47) TSHRNUDT1LMNACYP1A2HTT
SCHEMBL14595394 0.70 CHRM4 (0.58) MAPK1ALDH1A1CLK4HIF1ACYP2C19
SCHEMBL8646161 0.70 EGFR (0.48) EGFRMAPK1ALDH1A1CLK4HIF1A
SCHEMBL13351953 0.69 PIK3CD (0.39) EGFRCSF1RNUDT1LMNAHTT
SCHEMBL10072172 0.68 KDM4E (0.64) MAPK1ALDH1A1CLK4HIF1ACYP2C19
SCHEMBL2918443 0.67 HTT (0.70) MAPK1ALDH1A1CLK4CYP2C19TSHR
SCHEMBL24201767 0.67 PIK3CD (0.35) MAPK1ALDH1A1HIF1ALMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012055466-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-05-03 WO disclosed