SCHEMBL10074010

SCHEMBL10074010

COc1ccc([C@H]2c3ccc(O)c(C)c3OC[C@H]2c2ccc(O)cc2)cc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 4/20 0.39
CYP2D6 P10635 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
MAPK1 P28482 1/20 0.36
PPARG P37231 3/20 0.36
PPARD Q03181 3/20 0.36
ALOX5 P09917 1/20 0.36
PTPN1 P18031 1/20 0.36
TUBB4A P04350 3/20 0.35
TUBB P07437 3/20 0.35
TUBA3C P0DPH7 3/20 0.35
TUBA1B P68363 3/20 0.35
TUBA4A P68366 3/20 0.35
TUBB4B P68371 3/20 0.35
TUBB3 Q13509 3/20 0.35
TUBB2A Q13885 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362778 1.00 PTGS1 (0.41) PTGS1MEN1KMT2ACYP3A4CYP2D6
SCHEMBL15312110 1.00 PTGS1 (0.41) PTGS1MEN1KMT2ACYP3A4CYP2D6
SCHEMBL2713457 1.00 PTGS1 (0.41) PTGS1MEN1KMT2ACYP3A4CYP2D6
SCHEMBL15965355 0.93 PTGS1 (0.41) PTGS1MEN1KMT2ACYP3A4CYP2D6
SCHEMBL30362814 0.90 ESR1 (0.36) PTGS1CYP3A4CYP2D6PTPN1
SCHEMBL10074001 0.90 ESR1 (0.36) PTGS1CYP3A4CYP2D6PTPN1
SCHEMBL2713088 0.90 ESR1 (0.36) PTGS1CYP3A4CYP2D6PTPN1
SCHEMBL15312086 0.90 ESR1 (0.36) PTGS1CYP3A4CYP2D6PTPN1
SCHEMBL2716699 0.89 KDM1A (0.41) PTGS1CYP3A4CYP2D6MAOAMAOB
SCHEMBL10098035 0.89 KDM1A (0.41) PTGS1CYP3A4CYP2D6MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12414934-B2 Combination therapies Aardvark Therapeutics, Inc. (US) 2025-09-16 US disclosed
US-12329739-B2 Isoflavonoid compounds and methods for the treatment of cancer Aardvark Therapeutic, Inc. (US) 2025-06-17 US disclosed
US-12318364-B2 Isoflavonoid compositions and methods for the treatment of cancer Aardvark Therapeutics, Inc. (US) 2025-06-03 US disclosed
WO-2024137472-A2 COMBINATION THERAPIES MEI PHARMA, INC. (US) 2024-06-27 WO disclosed
US-20240165073-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER Aardvark Therapeutics, Inc. 2024-05-23 US disclosed
US-20230372287-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER Aardvark Therapeutics, Inc. 2023-11-23 US disclosed
US-20230372287-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER Aardvark Therapeutics, Inc. 2023-11-23 US disclosed
US-20230372287-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER Aardvark Therapeutics, Inc. 2023-11-23 US disclosed
US-11723893-B2 Isoflavonoid compositions and methods for the treatment of cancer MEI PHARMA, INC. (US) 2023-08-15 US disclosed
US-11723893-B2 Isoflavonoid compositions and methods for the treatment of cancer MEI PHARMA, INC. (US) 2023-08-15 US disclosed
US-9708283-B2 Isoflavonoid compositions and methods for the treatment of cancer MEI PHARMA, INC. (US) 2017-07-18 US disclosed
US-9708283-B2 Isoflavonoid compositions and methods for the treatment of cancer MEI PHARMA, INC. (US) 2017-07-18 US disclosed
US-9663484-B2 Isoflavonoid compounds and methods for the treatment of cancer MEI PHARMA, INC. (US) 2017-05-30 US disclosed
US-9663484-B2 Isoflavonoid compounds and methods for the treatment of cancer MEI PHARMA, INC. (US) 2017-05-30 US disclosed
US-20140234295-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2014-08-21 US disclosed
US-20140234295-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2014-08-21 US disclosed
US-20130273177-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2013-10-17 US disclosed
US-20130273177-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2013-10-17 US disclosed
WO-2012061409-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2012-05-10 WO disclosed
WO-2012061413-A2 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER MARSHALL EDWARDS, INC. (US) 2012-05-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12414934-B2 Combination therapies PCK2, PDK1, PCK1 PTGS1 1926/4885MEN1 4343/4885KMT2A 1455/4885
US-11723893-B2 Isoflavonoid compositions and methods for the treatment of cancer BAX, CASP3, SI PTGS1 1103/4885MEN1 4303/4885KMT2A 4470/4885
US-20240165073-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER BAX, CASP3, SI PTGS1 1103/4885MEN1 4303/4885KMT2A 4470/4885
US-20130273177-A1 ISOFLAVONOID COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER BAX, CASP3, SI PTGS1 1103/4885MEN1 4303/4885KMT2A 4470/4885
US-12318364-B2 Isoflavonoid compositions and methods for the treatment of cancer BAX, CASP3, SI PTGS1 1103/4885MEN1 4303/4885KMT2A 4470/4885
US-20140234295-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER BAX, CASP3, API5 PTGS1 326/4885MEN1 4218/4885KMT2A 3410/4885
US-20230372287-A1 ISOFLAVONOID COMPOUNDS AND METHODS FOR THE TREATMENT OF CANCER BAX, CASP3, API5 PTGS1 326/4885MEN1 4218/4885KMT2A 3410/4885
US-12329739-B2 Isoflavonoid compounds and methods for the treatment of cancer BAX, CASP3, API5 PTGS1 326/4885MEN1 4218/4885KMT2A 3410/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.