SCHEMBL10076865

SCHEMBL10076865

CC(=O)C(=O)SC(C)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
ALOX5 P09917 1/20 0.43
CYP2D6 P10635 1/20 0.40
SRC P12931 1/20 0.40
LMNA P02545 2/20 0.39
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
RECQL P46063 1/20 0.38
MAPT P10636 1/20 0.38
DAO P14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28340407 0.86 CYP2D6 (0.41) ALOX5CYP2D6SRCLMNACES2
SCHEMBL1959777 0.83 TSHR (0.46) HPGDALOX5CYP2D6SRCLMNA
SCHEMBL27838181 0.76 GPR139 (0.49) HPGDCYP2D6SRCLMNACES2
SCHEMBL14355132 0.75 HPGD (0.42) HPGDCYP2D6LMNAKMT2ADAO
SCHEMBL14355125 0.75 ADRA2C (0.39) CYP2D6LMNAKMT2ADAO
SCHEMBL12590975 0.75 ADRA2C (0.39) CYP2D6LMNAKMT2ADAO
SCHEMBL9817188 0.73 CYP2C19 (0.41) HPGDALOX5CYP2D6SRCLMNA
SCHEMBL11443376 0.72 ADRA2C (0.40) CYP2D6LMNAKMT2ADAO
SCHEMBL6535241 0.72 ADRA2C (0.40) CYP2D6LMNAKMT2ADAO
SCHEMBL3929030 0.72 POLB (0.44) HPGDLMNACES2CES1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468744-A2 Inhibitors of serine proteases, particularly HCV NS3-NS4A protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-27 EP disclosed