SCHEMBL10078853

SCHEMBL10078853

CN(CC(=O)O)C(=O)c1ccc(N)c(N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPT P10636 3/20 0.41
GAA P10253 3/20 0.41
MAPK1 P28482 1/20 0.41
ITGB3 P05106 2/20 0.40
ITGA2B P08514 2/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
HPGD P15428 4/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
GFER P55789 1/20 0.37
PLEC Q15149 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12010059 0.86 ALDH1A1 (0.46) MEN1KMT2AITGB3ITGA2BPDK1
SCHEMBL4027372 0.83 PDK1 (0.39) MEN1KMT2AMAPK1ITGB3ITGA2B
SCHEMBL11107022 0.82 HDAC1 (0.45) MEN1KMT2AMAPTITGB3ITGA2B
SCHEMBL24722155 0.81 MAPT (0.44) MAPTMAPK1ITGB3ITGA2BALDH1A1
SCHEMBL6865515 0.78 MAPT (0.48) MAPTGAAMAPK1PDK2HPGD
SCHEMBL12302105 0.75 KMT2A (0.48) MEN1KMT2AALDH1A1
SCHEMBL27622304 0.75 PIN1 (0.35) MEN1KMT2AITGB3ITGA2BPDK1
SCHEMBL4029711 0.75 PIN1 (0.35) MEN1KMT2AITGB3ITGA2BPDK1
SCHEMBL2282162 0.74 KMT2A (0.53) MEN1KMT2AHPGDALDH1A1PIN1
SCHEMBL4223718 0.74 P2RX7 (0.51) MAPTHPGDALDH1A1HTTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1789039-B1 S-TRIAZOLYL ALPHA -MERCAPTOACETANILDES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE ARDEA BIOSCIENCES INC (US) 2012-01-11 EP disclosed