SCHEMBL10085303

SCHEMBL10085303

COP(=O)(NCCCCN(C)C)OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
ALDH1A1 P00352 1/20 0.39
PAOX Q6QHF9 1/20 0.34
DNM1 Q05193 3/20 0.33
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4A O75164 5/20 0.30
KDM4C Q9H3R0 5/20 0.30
ANPEP P15144 1/20 0.30
KDM5A P29375 1/20 0.30
KDM7A Q6ZMT4 1/20 0.30
PHF8 Q9UPP1 1/20 0.30
KDM2A Q9Y2K7 1/20 0.30
PRMT3 O60678 1/20 0.30
CARM1 Q86X55 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15150904 0.94 TDP1 (0.38) TSHRALDH1A1PAOXDNM1TDP1
SCHEMBL15786625 0.89 ALDH1A1 (0.33) TSHRALDH1A1PAOX
SCHEMBL15150882 0.85 PRMT3 (0.39) ALDH1A1DNM1TDP1CYP2C9CYP2C19
SCHEMBL15786595 0.83 TDP1 (0.33) TSHRALDH1A1PAOXDNM1TDP1
SCHEMBL15028245 0.82 TSHR (0.37) TSHRALDH1A1PAOXDNM1TDP1
SCHEMBL10081267 0.79 ALDH1A1 (0.34) TSHRALDH1A1PAOXDNM1ANPEP
SCHEMBL24172211 0.79 TDP1 (0.39) TSHRALDH1A1PAOXDNM1TDP1
SCHEMBL15028248 0.76 TDP1 (0.36) TSHRALDH1A1PAOXDNM1TDP1
SCHEMBL24268008 0.75 PAOX (0.38) TSHRPAOXCYP2C9CYP2C19MEN1
SCHEMBL28932747 0.75 EPHX1 (0.45) TSHRALDH1A1ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303598-A1 BIOINSPIRED LIPID DERIVATIVES AND USES THEREOF OHIO STATE INNOVATION FOUNDATION 2023-09-28 US disclosed
EP-3860561-B1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS ALNYLAM PHARMACEUTICALS INC (US) 2023-06-21 EP disclosed
WO-2022040310-A2 BIOINSPIRED LIPID DERIVATIVES AND USES THEREOF OHIO STATE INNOVATION FOUNDATION (US) 2022-02-24 WO disclosed
WO-2022002040-A1 LIPID COMPOUNDS AND LIPID NANOPARTICLE COMPOSITIONS Suzhou Abogen Biosciences Co., Ltd. (CN) 2022-01-06 WO disclosed
US-9687448-B2 Nucleic acid lipid particle formulations ALNYLAM PHARMACEUTICALS, INC. (US) 2017-06-27 US disclosed
US-9682922-B2 Biodegradable lipids for the delivery of active agents ALNYLAM PHARMACEUTICALS, INC. (US) 2017-06-20 US disclosed
US-9463247-B2 Branched alkyl and cycloalkyl terminated biodegradable lipids for the delivery of active agents ALNYLAM PHARMACEUTICALS, INC. (US) 2016-10-11 US disclosed
US-20160009637-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS BANK OF AMERICA, N.A. 2016-01-14 US disclosed
US-20150306039-A1 IMPROVED NUCLEIC ACID LIPID PARTICLE FORMULATIONS BANK OF AMERICA, N.A. 2015-10-29 US disclosed
US-20150273068-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS BANK OF AMERICA, N.A. 2015-10-01 US disclosed
US-9061063-B2 Biodegradable lipids for the delivery of active agents ALNYLAM PHARMACEUTICALS, INC. (US) 2015-06-23 US disclosed
US-9012498-B2 Biodegradable lipids for the delivery of active agents ALNYLAM PHARMACEUTICALS, INC. (US) 2015-04-21 US disclosed
US-20150005363-A1 Branched Alkyl And Cycloalkyl Terminated Biodegradable Lipids For The Delivery Of Active Agents BANK OF AMERICA, N.A. 2015-01-01 US disclosed
US-20130195920-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS ALNYLAM PHARMACEUTICALS, INC. (US) 2013-08-01 US disclosed
US-20120027803-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS ALNYLAM PHARMACEUTICALS, INC. (US) 2012-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150005363-A1 Branched Alkyl And Cycloalkyl Terminated Biodegradable Lipids For The Delivery Of Active Agents LIPA, CETP, APOB TSHR 2909/4885ALDH1A1 1852/4885PAOX 352/4885
US-20120027803-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS LIPA, CETP, APOB TSHR 2854/4885ALDH1A1 2749/4885PAOX 524/4885
US-20160009637-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS LIPA, CETP, APOB TSHR 2854/4885ALDH1A1 2749/4885PAOX 524/4885
US-20230303598-A1 BIOINSPIRED LIPID DERIVATIVES AND USES THEREOF LIPA, APOB, LIPG TSHR 4293/4885ALDH1A1 1246/4885PAOX 1520/4885
US-20130195920-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS LIPA, APOB, CETP TSHR 2733/4885ALDH1A1 3151/4885PAOX 651/4885
US-20150273068-A1 BIODEGRADABLE LIPIDS FOR THE DELIVERY OF ACTIVE AGENTS LIPA, APOB, CETP TSHR 2733/4885ALDH1A1 3151/4885PAOX 651/4885
US-20150306039-A1 IMPROVED NUCLEIC ACID LIPID PARTICLE FORMULATIONS LIPA, NPC1L1, CETP TSHR 3683/4885ALDH1A1 2297/4885PAOX 812/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.