SCHEMBL10102822

SCHEMBL10102822

COc1cc(F)c(C(C)C)cc1BO

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.36
P2RX2 Q9UBL9 1/20 0.36
GAA P10253 2/20 0.34
POLB P06746 1/20 0.34
GFER P55789 1/20 0.34
CETP P11597 1/20 0.33
EIF4A3 P38919 1/20 0.33
MGAM O43451 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
KCNK3 O14649 1/20 0.30
KCNK9 Q9NPC2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10077746 0.84 P2RX3 (0.37) P2RX3P2RX2GAAPOLBGFER
SCHEMBL19650317 0.84 GAA (0.44) P2RX3P2RX2GAAPOLBGFER
SCHEMBL23288682 0.79 THRB (0.37) P2RX3P2RX2GAAPOLBGFER
SCHEMBL5166833 0.79 P2RX3 (0.45) P2RX3P2RX2GAAPOLBGFER
SCHEMBL15927601 0.78 P2RX3 (0.41) P2RX3P2RX2GAAPOLBGFER
SCHEMBL13059718 0.77 GAA (0.48) P2RX3P2RX2GAAPOLBGFER
SCHEMBL12190518 0.77 P2RX3 (0.48) P2RX3P2RX2GAAPOLBGFER
SCHEMBL22781546 0.77 TUBB1 (0.34) LMNAMAPK1HTTRAB9A
SCHEMBL24449860 0.77 ALOX15 (0.40) P2RX3P2RX2GAAPOLBGFER
SCHEMBL18387027 0.76 CETP (0.31) P2RX3P2RX2CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2468735-A1 Synthesis of intermediates for preparing anacetrapib and derivates thereof LEK Pharmaceuticals d.d. (SI) 2012-06-27 EP disclosed