SCHEMBL1011352

SCHEMBL1011352

COc1ccccc1Oc1cnc(-c2nccc(Cl)n2)nc1Cl

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
DHPS P49366 12/20 0.43
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PIN1 Q13526 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700406 0.90 LMNA (0.50) LMNADHPSKMT2AMEN1POLB
SCHEMBL625229 0.78 CYP1A2 (0.44) LMNAKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL1443043 0.76 LMNA (0.44) LMNAKMT2AMEN1POLBL3MBTL1
SCHEMBL13674052 0.75 CYP1A2 (0.63) LMNAKMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL14483989 0.74 KMT2A (0.56) LMNAKMT2AMEN1POLBL3MBTL1
SCHEMBL29770374 0.73 DHPS (0.58) DHPS
SCHEMBL618135 0.73 DHPS (0.58) DHPS
SCHEMBL1011353 0.72 LMNA (0.46) LMNADHPSKMT2AMEN1POLB
SCHEMBL2071241 0.70 KMT2A (0.68) LMNADHPSKMT2AMEN1POLB
SCHEMBL1442223 0.70 LMNA (0.67) LMNAKMT2AMEN1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268634-A2 PROCESSES FOR THE PREPARATION OF BOSENTAN AND RELATED COMPOUNDS USING NOVEL INTERMEDIATES Actavis Group PTC EHF (IS) 2011-01-05 EP disclosed
WO-2009112954-A2 PROCESSES FOR THE PREPARATION OF BOSENTAN AND RELATED COMPOUNDS USING NOVEL INTERMEDIATES ACTAVIS GROUP PTC EHF (IS) 2009-09-17 WO disclosed