SCHEMBL10117537

SCHEMBL10117537

CCCCNC(=O)Nc1ncc(-c2ccc(Br)cc2)n1C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.38
HTT P42858 2/20 0.38
MGLL Q99685 1/20 0.38
EPHX2 P34913 1/20 0.38
NR1H2 P55055 1/20 0.37
P2RY1 P47900 1/20 0.37
ATM Q13315 1/20 0.36
PDE5A O76074 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE1C Q14123 1/20 0.36
PDE3A Q14432 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10117508 0.94 NPC1 (0.41) RAB9ANPC1SMN1; SMN2NR1H2IDO1
SCHEMBL10117536 0.90 MTOR (0.38) NR1H2IDO1GAA
SCHEMBL10117540 0.85 NR1H2 (0.49) RAB9ANPC1NR1H2KDM4EHDAC8
SCHEMBL10117510 0.84 MEN1 (0.45) RAB9ANPC1SMN1; SMN2NR1H2ALDH1A1
SCHEMBL10117499 0.82 FPR2 (0.39) RAB9ANPC1SMN1; SMN2HTTNR1H2
SCHEMBL10117881 0.78 MAPK1 (0.43) SMN1; SMN2ALDH1A1
SCHEMBL4242529 0.75 GABRG2 (0.38) RAB9ANPC1SMN1; SMN2NR1H2ALDH1A1
SCHEMBL10117534 0.73 NR1H2 (0.40) NR1H2IDO1
SCHEMBL4298498 0.72 FFAR1 (0.39) NR1H2HDAC3HDAC1HDAC2HDAC8
SCHEMBL4231082 0.72 NR1H2 (0.41) RAB9ANPC1SMN1; SMN2NR1H2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087976-A2 NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-06-28 WO disclosed