SCHEMBL10119347

SCHEMBL10119347

Cc1cccc(-c2cccnc2C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4)cc3)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GAA P10253 2/20 0.40
DHODH Q02127 3/20 0.39
SCN9A Q15858 2/20 0.37
ROCK2 O75116 2/20 0.37
KHK P50053 1/20 0.37
SCN3A Q9NY46 2/20 0.37
HCRTR1 O43613 2/20 0.37
PFKFB2 O60825 1/20 0.37
PFKFB1 P16118 1/20 0.37
PFKFB3 Q16875 1/20 0.37
HCRTR2 O43614 1/20 0.37
KMT2A Q03164 1/20 0.36
PDGFRB P09619 2/20 0.36
FLT3 P36888 2/20 0.36
IKBKB O14920 1/20 0.36
JAK2 O60674 1/20 0.36
KIT P10721 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845640 0.92 ALDH1A1 (0.49) ALDH1A1TSHRNPSR1GAAROCK2
SCHEMBL10119326 0.91 EP300 (0.41) ALDH1A1SCN9AROCK2SCN3APDGFRB
SCHEMBL10119342 0.88 ALDH1A1 (0.45) ALDH1A1TSHRNPSR1GAAHCRTR1
SCHEMBL845114 0.83 EP300 (0.46) ALDH1A1
SCHEMBL845841 0.82 TRPV1 (0.45) ALDH1A1ROCK2HCRTR1HCRTR2
SCHEMBL13272509 0.82 TRPV1 (0.45) ALDH1A1ROCK2HCRTR1HCRTR2
SCHEMBL10119551 0.82 DHODH (0.40) ALDH1A1GAADHODHSCN9AROCK2
SCHEMBL845374 0.81 PABPC1 (0.51) ALDH1A1TSHRNPSR1GAAROCK2
SCHEMBL872415 0.81 PABPC1 (0.38) ALDH1A1GAASCN9AROCK2SCN3A
SCHEMBL871971 0.81 PDE5A (0.42) GAASCN9AROCK2SCN3AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed