SCHEMBL871971

SCHEMBL871971

CCCOc1cccnc1C(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.42
GAA P10253 1/20 0.41
PABPC1 P11940 1/20 0.40
HSD17B10 Q99714 1/20 0.39
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
SCN9A Q15858 2/20 0.37
SCN3A Q9NY46 2/20 0.37
SCN5A Q14524 1/20 0.37
PFKFB3 Q16875 4/20 0.37
PFKFB2 O60825 3/20 0.37
PFKFB1 P16118 3/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ROCK2 O75116 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845330 0.92 GAA (0.47) PDE5AGAAPABPC1LMNAKDM4E
SCHEMBL872415 0.86 PABPC1 (0.38) GAAPABPC1LMNAKDM4EMAPK1
SCHEMBL871771 0.83 PABPC1 (0.44) GAAPABPC1LMNAKDM4EMAPK1
SCHEMBL872930 0.82 GAA (0.52) GAAPABPC1LMNAKDM4EMAPK1
SCHEMBL10119551 0.82 DHODH (0.40) GAASCN9ASCN3ASCN5ACYP2C9
SCHEMBL10119636 0.81 CYP2C9 (0.38) PABPC1MAPK1SCN9ASCN3APFKFB3
SCHEMBL10119347 0.81 ALDH1A1 (0.43) GAASCN9ASCN3APFKFB3PFKFB2
SCHEMBL10119513 0.80 JAK2 (0.41) SCN9ASCN3ASCN5ACYP2C9CYP2C19
SCHEMBL845060 0.80 KDM4E (0.51) GAAPABPC1HSD17B10LMNAKDM4E
SCHEMBL845518 0.80 GAA (0.52) PDE5AGAAPABPC1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed