SCHEMBL10119595

SCHEMBL10119595

CC(C)(C)CON1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN3A Q9NY46 3/20 0.43
SCN9A Q15858 3/20 0.43
SCN5A Q14524 1/20 0.43
PSMB8 P28062 2/20 0.40
HDAC8 Q9BY41 2/20 0.39
PFKFB3 Q16875 7/20 0.39
PFKFB1 P16118 6/20 0.39
PFKFB2 O60825 5/20 0.39
DPP4 P27487 3/20 0.39
DPP8 Q6V1X1 1/20 0.39
NPC1 O15118 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873304 0.87 PFKFB3 (0.39) SCN3ASCN9ASCN5APSMB8HDAC8
SCHEMBL873706 0.84 PFKFB2 (0.42) SCN3ASCN9AHDAC8PFKFB3PFKFB1
SCHEMBL872815 0.83 PSMB8 (0.38) SCN3ASCN9ASCN5APSMB8HDAC8
SCHEMBL871886 0.82 SCN3A (0.39) SCN3ASCN9ASCN5APSMB8HDAC8
SCHEMBL844873 0.81 NPC1 (0.63) SCN3ASCN9ASCN5AHDAC8DPP4
SCHEMBL872886 0.80 KDM4E (0.52) PFKFB3PFKFB1PFKFB2NPC1
SCHEMBL10119687 0.79 CYP2C9 (0.44) PSMB8HDAC8PFKFB3PFKFB1PFKFB2
SCHEMBL845510 0.79 SCN3A (0.54) SCN3ASCN9ASCN5APSMB8HDAC8
SCHEMBL10119593 0.76 NPC1 (0.51) SCN3ASCN9ASCN5AHDAC8DPP4
SCHEMBL845110 0.75 ALDH1A1 (0.48) PFKFB3PFKFB1PFKFB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed