SCHEMBL872815

SCHEMBL872815

Cn1cccc1CON1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 1/20 0.38
HDAC8 Q9BY41 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
PFKFB3 Q16875 11/20 0.37
PFKFB1 P16118 10/20 0.37
PFKFB2 O60825 8/20 0.37
SCN3A Q9NY46 3/20 0.36
SCN9A Q15858 2/20 0.36
SCN5A Q14524 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
KHK P50053 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10119595 0.83 SCN3A (0.43) PSMB8HDAC8HDAC3HDAC4HDAC1
SCHEMBL873304 0.82 PFKFB3 (0.39) PSMB8HDAC8HDAC3HDAC4HDAC1
SCHEMBL873706 0.80 PFKFB2 (0.42) HDAC8HDAC3HDAC4HDAC1HDAC7
SCHEMBL871886 0.77 SCN3A (0.39) PSMB8HDAC8HDAC3HDAC4HDAC1
SCHEMBL872886 0.75 KDM4E (0.52) PFKFB3PFKFB1PFKFB2
SCHEMBL845237 0.74 ALDH1A1 (0.45)
SCHEMBL10119687 0.74 CYP2C9 (0.44) PSMB8HDAC8PFKFB3PFKFB1PFKFB2
SCHEMBL845510 0.74 SCN3A (0.54) PSMB8HDAC8HDAC3HDAC4HDAC1
SCHEMBL844873 0.73 NPC1 (0.63) HDAC8SCN3ASCN9ASCN5A
SCHEMBL845110 0.72 ALDH1A1 (0.48) PFKFB3PFKFB1PFKFB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed