SCHEMBL10120030

SCHEMBL10120030

Cc1n[nH]c2c(N)ncnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 4/20 0.44
PI4K2B Q8TCG2 4/20 0.44
PI4K2A Q9BTU6 4/20 0.44
PI4KB Q9UBF8 4/20 0.44
XDH P47989 2/20 0.44
LRRK2 Q5S007 2/20 0.44
LMNA P02545 1/20 0.44
DRD3 P35462 1/20 0.44
PDPK1 O15530 1/20 0.43
LIMK1 P53667 2/20 0.41
ERAP1 Q9NZ08 1/20 0.39
PIK3CD O00329 2/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
PRKDC P78527 2/20 0.38
NUDT1 P36639 2/20 0.37
CDC7 O00311 2/20 0.37
DBF4 Q9UBU7 2/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24121974 0.83 PDPK1 (0.46) PDPK1ADORA2ADYRK1AYTHDC1YTHDF2
SCHEMBL6155249 0.80 LIMK1 (0.44) PI4KAPI4K2BPI4K2API4KBXDH
Hydrochloric Acid SCHEMBL7166188 0.78 PI4KA (0.45) PI4KAPI4K2BPI4K2API4KBXDH
SCHEMBL11330441 0.78 PDPK1 (0.42) PDPK1ADORA2AYTHDC1YTHDF2ADORA2B
SCHEMBL3237641 0.78 KDM4E (0.42) LMNAPDPK1KDM4EALDH1A1MAPT
SCHEMBL3113393 0.75 LIMK1 (0.41) PI4KAPI4K2BPI4K2API4KBXDH
SCHEMBL30515894 0.75 LIMK1 (0.41) PI4KAPI4K2BPI4K2API4KBXDH
SCHEMBL11337092 0.75 TP53 (0.49) LMNAPDPK1CDC7DBF4ALDH1A1
SCHEMBL19402816 0.75 PIK3CD (0.38) PI4KAPI4K2BPI4K2API4KBXDH
SCHEMBL21539447 0.75 MTAP (0.39) PI4KAPI4K2BPI4K2API4KBXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113039182-B Inhibitors of YAP/TAZ-TEAD interactions and their use in cancer treatment 伊文蒂瓦公司 2024-02-20 CN claimed
WO-2025242872-A1 1H-PYRAZOLO[4,3-D]PYRIMIDINE DERIVATIVES Apollo AP45 Limited (GB) 2025-11-27 WO disclosed
CN-113039182-B Inhibitors of YAP/TAZ-TEAD interactions and their use in cancer treatment 伊文蒂瓦公司 2024-02-20 CN disclosed
US-20230181546-A1 TREATMENT OF RESPIRATORY DISEASES WITH AMINO ACID COMPOUNDS PLIANT THERAPEUTICS INC (US) 2023-06-15 US disclosed
WO-2022219636-A1 ANTI-VIRAL AND ANTI-TUMORAL COMPOUNDS, AND USES THEREOF YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2022-10-20 WO disclosed
EP-3083617-B1 ISOCHROMENE DERIVATIVES AS PHOSPHOINOSITIDE 3-KINASES INHIBITORS CHIESI FARM SPA (IT) 2019-09-11 EP disclosed
US-20170275322-A1 METHODS FOR THE PREPARATION OF DIASTEREOMERICALLY PURE PHOSPHORAMIDATE PRODRUGS MEDIVIR AB (SE) 2017-09-28 US disclosed
US-20170044206-A1 CYCLIC DI-NUCLEOTIDE COMPOUNDS AS STING AGONISTS MERCK SHARP & DOHME CORP. (US) 2017-02-16 US disclosed
US-9487544-B2 Methods for the preparation of diasteromerically pure phosphoramidate prodrugs GILEAD SCIENCES, INC. (US) 2016-11-08 US disclosed
EP-3083617-A1 ISOCHROMENE DERIVATIVES AS PHOSPHOINOSITIDE 3-KINASES INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2016-10-26 EP disclosed
US-8790919-B2 Compositions and methods for optimizing cleavage of RNA by RNase H ISIS PHARMACEUTICALS, INC. (US) 2014-07-29 US disclosed
US-20130281686-A1 METHODS FOR THE PREPARATION OF DIASTEROMERICALLY PURE PHOSPHORAMIDATE PRODRUGS GILEAD SCIENCES, INC. (US) 2013-10-24 US disclosed
WO-2012012465-A1 METHODS FOR THE PREPARATION OF DIASTEROMERICALLY PURE PHOSPHORAMIDATE PRODRUGS CLARKE, MICHAEL, O'NEIL HANRAHAN (US) 2012-01-26 WO disclosed
US-7939677-B2 Oligomeric compounds comprising 4′-thionucleosides for use in gene modulation ISIS PHARMACEUTICALS, INC. (US) 2011-05-10 US disclosed
US-20100324277-A1 OLIGOMERIC COMPOUNDS COMPRISING 4'-THIONUCLEOSIDES FOR USE IN GENE MODULATION ISIS PHARMACEUTICALS, INC. (US) 2010-12-23 US disclosed
US-7713944-B2 Oligomers comprising activated disulfides which bind to plasma proteins and their use for delivery to cells ISIS PHARMACEUTICALS, INC. (US) 2010-05-11 US disclosed
US-20080293666-A1 Antibacterial Agents REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2008-11-27 US disclosed
US-20080207541-A1 Contacting a eukaryotic cell with a mixed backbone oligonucleotide with a first region that forms a substrate for cleavage by an RNase and a second region which does not, and a transition moiety which modulates the transmission of the conformation of said second region into the first region IONIS PHARMACEUTICALS, INC. 2008-08-28 US disclosed
US-7368437-B1 Bicyclic heterocycles, processes for their preparation and their use as herbicides and pharmaceutical agents BAYER CROPSCIENCE AG (DE) 2008-05-06 US disclosed
US-20070276139-A1 Substituted Pixyl Protecting Groups for Oligonucleotide Synthesis ISIS PHARMACEUTICALS, INC. 2007-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080207541-A1 Contacting a eukaryotic cell with a mixed backbone oligonucleotide with a first region that forms a substrate for cleavage by an RNase and a second region which does not, and a transition moiety which modulates the transmission of the conformation of said second region into the first region RNASEH1, NSUN3, RNASEL PI4KA 3085/4885PI4K2B 2693/4885PI4K2A 2841/4885
US-20130281686-A1 METHODS FOR THE PREPARATION OF DIASTEROMERICALLY PURE PHOSPHORAMIDATE PRODRUGS PAICS, DPYD, PNP PI4KA 787/4885PI4K2B 728/4885PI4K2A 961/4885
US-20170275322-A1 METHODS FOR THE PREPARATION OF DIASTEREOMERICALLY PURE PHOSPHORAMIDATE PRODRUGS PNP, PAICS, NUDT1 PI4KA 769/4885PI4K2B 1232/4885PI4K2A 1162/4885
US-20100324277-A1 OLIGOMERIC COMPOUNDS COMPRISING 4'-THIONUCLEOSIDES FOR USE IN GENE MODULATION SNRPE, NSUN3, NSUN2 PI4KA 1842/4885PI4K2B 1405/4885PI4K2A 1416/4885
US-20170044206-A1 CYCLIC DI-NUCLEOTIDE COMPOUNDS AS STING AGONISTS STING1, CGAS, IFNAR1 PI4KA 2270/4885PI4K2B 1878/4885PI4K2A 1358/4885
US-20070276139-A1 Substituted Pixyl Protecting Groups for Oligonucleotide Synthesis RPP30, NOP10, NR0B1 PI4KA 3369/4885PI4K2B 2362/4885PI4K2A 2480/4885
US-20080293666-A1 Antibacterial Agents MRPL21, ABCB7, MSR1 PI4KA 4490/4885PI4K2B 3867/4885PI4K2A 4444/4885
US-20230181546-A1 TREATMENT OF RESPIRATORY DISEASES WITH AMINO ACID COMPOUNDS ITGA5, ITGAL, ITGB5 PI4KA 2340/4885PI4K2B 3355/4885PI4K2A 3173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.