SCHEMBL10120532

SCHEMBL10120532

COC(=O)c1cc(-n2cc(-c3ccc(Cl)c(Cl)c3)nn2)c2ccccc2n1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.42
POLB P06746 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
BCHE P06276 1/20 0.40
HTT P42858 1/20 0.40
KMO O15229 3/20 0.40
ABCG2 Q9UNQ0 3/20 0.40
DHODH Q02127 1/20 0.40
CDC7 O00311 1/20 0.40
OGT O15294 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1695207 0.89 KMO (0.51) POLBMEN1CYP1A2CYP2D6MAPT
SCHEMBL10120527 0.89 ABCG2 (0.46) KDM4EMEN1KMT2ABCHEABCG2
SCHEMBL1694845 0.82 KDM4E (0.51) POLBKDM4EMEN1CYP1A2CYP2D6
SCHEMBL1694435 0.77 OGT (0.45) NOTUMKDM4EABCG2DHODHOGT
SCHEMBL1694971 0.76 LDHA (0.53) KDM4EBCHEKMOABCG2DHODH
SCHEMBL15100599 0.74 DHODH (0.47) POLBKDM4EMEN1CYP1A2CYP2D6
SCHEMBL3281879 0.72 KDM4E (0.60) POLBKDM4EMEN1MAPTKMT2A
SCHEMBL21044565 0.72 OGT (0.53) NOTUMKDM4EABCG2OGT
SCHEMBL15100471 0.70 PRSS12 (0.47) POLBKMODHODHCDC7OGT
SCHEMBL1939020 0.70 KMO (0.72) NOTUMKDM4EMAPTKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006068-A2 COMPOUNDS FOR THE INHIBITION OF CELLULAR PROLIFERATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-12 WO disclosed