SCHEMBL1014096

SCHEMBL1014096

CCCSc1ncc(C(=O)O)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HSD17B10 Q99714 2/20 0.44
ALOX15 P16050 1/20 0.44
HCAR3 P49019 8/20 0.42
MAPT P10636 1/20 0.42
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
P4HA1 P13674 1/20 0.38
P4HTM Q9NXG6 1/20 0.38
HCAR2 Q8TDS4 2/20 0.38
KDM6B O15054 1/20 0.38
KDM4A O75164 1/20 0.38
KDM4D Q6B0I6 1/20 0.38
KDM3B Q7LBC6 1/20 0.38
HIF1AN Q9NWT6 1/20 0.38
KDM5B Q9UGL1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28511099 0.88 KDM6B (0.50) KDM4EALDH1A1HSD17B10ALOX15HCAR3
SCHEMBL6302512 0.85 ALDH1A1 (0.47) KDM4EALDH1A1HSD17B10ALOX15HCAR3
SCHEMBL5660785 0.83 ALDH1A1 (0.41) KDM4EALDH1A1HSD17B10ALOX15HCAR3
SCHEMBL27884460 0.77 HCAR3 (0.49) KDM4EALDH1A1HSD17B10ALOX15HCAR3
SCHEMBL1015456 0.75 RAB9A (0.45) ALDH1A1HSD17B10MAPTCYP1A2CYP2C9
SCHEMBL19243077 0.74 KDM4E (0.42) KDM4EALDH1A1HSD17B10MAPTHPGD
SCHEMBL240773 0.74 ALDH1A1 (0.52) KDM4EALDH1A1HSD17B10ALOX15HCAR3
Ammonia Solution, Strong SCHEMBL28006349 0.74 ALDH1A1 (0.52) KDM4EALDH1A1HSD17B10ALOX15HCAR3
SCHEMBL5387520 0.73 ADORA3 (0.36) KDM4EMAPTADORA3SMN1; SMN2
SCHEMBL5387528 0.73 ADORA3 (0.36) KDM4EMAPTADORA3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271629-A1 SUBSTITUTED PYRIMIDIN-5-CARBOXAMIDES 281 AstraZeneca AB (SE) 2011-01-12 EP disclosed