SCHEMBL10145939

SCHEMBL10145939

CC(c1cccc(C(F)(F)F)c1)n1c(=O)n(C)c2cc(-c3ccccc3N)ccc21

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 7/20 0.38
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.38
MAPK14 Q16539 3/20 0.36
KRAS P01116 3/20 0.36
SOS1 Q07889 3/20 0.36
HSD17B2 P37059 1/20 0.36
ADORA2A P29274 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14992603 0.85 AR (0.45) KCNN4DRD3KCNH2MAPK14AR
SCHEMBL10146326 0.79 PIK3CA (0.42) MAPK14ADORA2A
SCHEMBL10145950 0.74 MAPK14 (0.53) MAPK14
SCHEMBL14992236 0.70 AR (0.47) MAPK14AR
SCHEMBL10146676 0.69 GRM2 (0.47) MAPK14
SCHEMBL398678 0.68 ADORA2A (0.54) ADORA2A
SCHEMBL10146672 0.67 PARG (0.46) MAPK14ADORA2A
SCHEMBL10146668 0.67 GRM2 (0.70)
SCHEMBL10145948 0.67 GRM2 (0.49) MAPK14ADORA2A
SCHEMBL10145941 0.65 GRM2 (0.47) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed