SCHEMBL10145950

SCHEMBL10145950

Cn1c(=O)n(C)c2cc(-c3ccccc3N)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.53
ATAD2 Q6PL18 1/20 0.46
ALDH1A1 P00352 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
GLA P06280 1/20 0.45
CHEK1 O14757 1/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
BRD4 O60885 1/20 0.45
BRPF1 P55201 1/20 0.45
CREBBP Q92793 1/20 0.44
GRM2 Q14416 1/20 0.43
BRD1 O95696 1/20 0.43
METAP2 P50579 1/20 0.43
S100B P04271 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.41
LMNA P02545 1/20 0.41
PKM P14618 1/20 0.41
TRIM24 O15164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10146672 0.86 PARG (0.46) MAPK14ATAD2ALDH1A1SMN1; SMN2GLA
SCHEMBL10145948 0.84 GRM2 (0.49) MAPK14CHEK1GRM2METAP2
SCHEMBL10146676 0.82 GRM2 (0.47) MAPK14ALDH1A1SMN1; SMN2CHEK1BRD4
SCHEMBL10146668 0.82 GRM2 (0.70) GRM2METAP2
SCHEMBL10145941 0.82 GRM2 (0.47) MAPK14ALDH1A1CHEK1GRM2METAP2
SCHEMBL10145952 0.80 GRM2 (0.45) MAPK14KDM4EGRM2METAP2MAPT
SCHEMBL10146004 0.79 BRD4 (0.48) ALDH1A1KDM4EBRD4GRM2MAPT
SCHEMBL10146671 0.79 PARG (0.51) MAPK14CHEK1GRM2METAP2
SCHEMBL14992133 0.77 MAPK14 (0.50) MAPK14ALDH1A1SMN1; SMN2GLAKDM4E
SCHEMBL10146326 0.77 PIK3CA (0.42) MAPK14ALDH1A1SMN1; SMN2HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed