SCHEMBL10146672

SCHEMBL10146672

Cn1c(=O)n(-c2ccccc2)c2ccc(-c3ccccc3N)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARG Q86W56 2/20 0.46
PGR P06401 1/20 0.44
MAPK14 Q16539 4/20 0.44
GRM2 Q14416 1/20 0.41
METAP2 P50579 1/20 0.41
CHEK1 O14757 1/20 0.40
GSK3B P49841 2/20 0.39
GSK3A P49840 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.37
GLA P06280 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPK1 P28482 1/20 0.36
ATAD2 Q6PL18 1/20 0.36
HSPA1A P0DMV8 1/20 0.36
PABPC1 P11940 1/20 0.36
CYP1A2 P05177 1/20 0.36
ADORA2A P29274 1/20 0.36
BRD1 O95696 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10145950 0.86 MAPK14 (0.53) MAPK14GRM2METAP2CHEK1ALDH1A1
SCHEMBL10146326 0.85 PIK3CA (0.42) MAPK14ALDH1A1HSD17B10MAPTSMN1; SMN2
SCHEMBL14993164 0.81 PARG (0.43) PARGPGRMAPK14GRM2ALDH1A1
SCHEMBL10145948 0.77 GRM2 (0.49) MAPK14GRM2METAP2CHEK1CYP1A2
SCHEMBL10145941 0.75 GRM2 (0.47) PGRMAPK14GRM2METAP2CHEK1
SCHEMBL10146676 0.75 GRM2 (0.47) PARGMAPK14GRM2METAP2CHEK1
SCHEMBL10146668 0.75 GRM2 (0.70) PARGGRM2METAP2
SCHEMBL15396477 0.75 PARG (0.43) PARGPGRMAPK14GRM2GSK3B
SCHEMBL15396697 0.75 PGR (0.50) PARGPGRMAPK14GRM2GSK3B
SCHEMBL6362809 0.74 PGR (0.68) PARGPGRGSK3BGSK3AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed