SCHEMBL10146676

SCHEMBL10146676

CC(C)Cn1c(=O)n(C)c2cc(-c3ccccc3N)ccc21

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.47
PARG Q86W56 1/20 0.45
ALDH1A1 P00352 1/20 0.45
BRD4 O60885 1/20 0.44
METAP2 P50579 2/20 0.41
AGER Q15109 1/20 0.40
HPD P32754 2/20 0.40
MAPK14 Q16539 2/20 0.39
PDE2A O00408 5/20 0.39
PDE1A P54750 5/20 0.39
PDE1B Q01064 5/20 0.39
PDE1C Q14123 5/20 0.39
CHEK1 O14757 1/20 0.38
LMNA P02545 1/20 0.38
STAT3 P40763 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SLC16A1 P53985 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10145948 0.85 GRM2 (0.49) GRM2METAP2HPDMAPK14CHEK1
SCHEMBL10145941 0.82 GRM2 (0.47) GRM2ALDH1A1METAP2HPDMAPK14
SCHEMBL10146668 0.82 GRM2 (0.70) GRM2PARGMETAP2
SCHEMBL10145950 0.82 MAPK14 (0.53) GRM2ALDH1A1BRD4METAP2MAPK14
SCHEMBL627494 0.82 GRM2 (0.44) GRM2PARGBRD4AGERHPD
SCHEMBL10145952 0.81 GRM2 (0.45) GRM2METAP2MAPK14
SCHEMBL10146004 0.80 BRD4 (0.48) GRM2PARGALDH1A1BRD4HPD
SCHEMBL10146671 0.80 PARG (0.51) GRM2PARGMETAP2MAPK14CHEK1
SCHEMBL8229445 0.76 AGER (0.62) PARGALDH1A1AGERHPDLMNA
SCHEMBL10146391 0.76 TRIM24 (0.40) GRM2PARGALDH1A1BRD4HPD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed