SCHEMBL10145973

SCHEMBL10145973

Cn1c(=O)n(C)c2cc(-c3cccc(N)c3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.48
GRM2 Q14416 1/20 0.48
BRD4 O60885 2/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 1/20 0.46
BRPF1 P55201 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MAOA P21397 2/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
ATAD2 Q6PL18 1/20 0.43
GLA P06280 1/20 0.43
MAOB P27338 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1843229 0.80 ALDH1A1 (0.56) BRD4ALDH1A1SMN1; SMN2KDM4EBRPF1
Ammonia Solution, Strong SCHEMBL1842927 0.78 ALDH1A1 (0.55) BRD4ALDH1A1SMN1; SMN2KDM4EBRPF1
Hydrochloric Acid SCHEMBL16736534 0.78 ALDH1A1 (0.55) BRD4ALDH1A1SMN1; SMN2KDM4EBRPF1
SCHEMBL10145950 0.75 MAPK14 (0.53) MAPK14GRM2BRD4ALDH1A1SMN1; SMN2
SCHEMBL768881 0.74 MAPK14 (0.58) MAPK14ALDH1A1
SCHEMBL15828332 0.71 PABPC1 (0.43) MAPK14BRD4ALDH1A1SMN1; SMN2KDM4E
SCHEMBL31131353 0.71 MAOA (0.84) ALDH1A1KDM4EHSD17B10MAOACA12
SCHEMBL29561461 0.71 MAOA (0.84) ALDH1A1KDM4EHSD17B10MAOACA12
SCHEMBL311194 0.71 MAOA (0.84) ALDH1A1KDM4EHSD17B10MAOACA12
Ethane SCHEMBL28815160 0.71 MAOA (0.75) ALDH1A1KDM4EMAOACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021382-A1 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2012-02-16 WO disclosed