SCHEMBL10151385

SCHEMBL10151385

COc1ccc2c(c1)nc(CF)n2-c1cnc(NC(=O)c2ccc(N=O)cc2F)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.36
RAB9A P51151 3/20 0.36
TP53 P04637 2/20 0.36
F10 P00742 2/20 0.36
MITF O75030 1/20 0.36
GAA P10253 1/20 0.36
KCNH2 Q12809 1/20 0.36
HPGDS O60760 1/20 0.35
PDE10A Q9Y233 1/20 0.34
BRD4 O60885 1/20 0.34
KMT2A Q03164 1/20 0.34
ROCK2 O75116 2/20 0.33
GRM5 P41594 1/20 0.33
ABCB1 P08183 1/20 0.33
ALDH1A1 P00352 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33
DYRK1A Q13627 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10151390 0.82 RAB9A (0.42) NPC1RAB9ATP53MITFGAA
SCHEMBL645754 0.79 HPGDS (0.40) NPC1RAB9ATP53F10MITF
SCHEMBL10239334 0.77 DEGS1 (0.43) NPC1RAB9ATP53HPGDSKMT2A
SCHEMBL647011 0.77 GRM5 (0.39) NPC1RAB9ATP53F10MITF
SCHEMBL10151672 0.77 RAB9A (0.44) NPC1RAB9AKMT2AGRM5KDM4E
SCHEMBL10151674 0.76 TP53 (0.38) NPC1RAB9ATP53MITFGAA
SCHEMBL648228 0.76 F10 (0.43) NPC1RAB9ATP53F10MITF
SCHEMBL645944 0.75 NPC1 (0.37) NPC1RAB9ATP53F10MITF
SCHEMBL645920 0.75 ORAI1 (0.45) NPC1RAB9ATP53MITFGAA
SCHEMBL646333 0.74 NPC1 (0.46) NPC1RAB9ATP53GAABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119643-B2 Benzoimidazolyl-pyrazine compounds for inflammation and immune-related uses SYNTA PHARMACEUTICALS CORP. (US) 2012-02-21 US disclosed