SCHEMBL10153305

SCHEMBL10153305

COC(=O)C1C(=O)N(OCc2ccccc2)C(=O)c2cc(Cl)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 1/20 0.46
POLB P06746 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.40
GAA P10253 1/20 0.40
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.37
PTGER1 P34995 2/20 0.37
S1PR1 P21453 1/20 0.37
S1PR5 Q9H228 1/20 0.37
TSHR P16473 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALDH2 P05091 1/20 0.37
ALDH3A1 P30838 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10154056 0.88 MEN1 (0.45) MEN1KMT2AMAPTPOLBCYP2C9
SCHEMBL9959325 0.88 APP (0.42) MEN1KMT2AMAPTALDH1A1
SCHEMBL9960564 0.87 TRPA1 (0.38) MEN1KMT2AMAPTALDH1A1
SCHEMBL10153698 0.87 ALDH1A1 (0.39) MEN1KMT2AMAPTCYP2C9GAA
SCHEMBL9959247 0.87 ALDH1A1 (0.42) MEN1KMT2AMAPTPOLBGAA
SCHEMBL9953482 0.87 MEN1 (0.48) MEN1KMT2AMAPTPOLBCYP2C9
SCHEMBL10153594 0.87 ACHE (0.45) MEN1KMT2AMAPTSMN1; SMN2PTGER1
SCHEMBL9958850 0.87 MEN1 (0.43) MEN1KMT2AMAPTPOLBCYP2C9
SCHEMBL10153293 0.85 ACHE (0.45) MEN1KMT2AMAPTPOLBSMN1; SMN2
SCHEMBL10153644 0.83 ALDH1A1 (0.42) MAPTCYP2C9L3MBTL1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed